Hrabinová Martina | Centrum biomedicínského výzkumu

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Hrabinová Martina

Info MH aj

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Postdoctoral fellow
hrabinovamartina@gmail.com
ORCID:0000-0002-9428-4109


Martina obtained her Master degree in 2014 in the study program Medical bioanalytics at the Faculty of Pharmacy in Hradec Kralove, Charles University in Prague. Currently, Martina is a student of doctoral degree program Toxicology at the Faculty of Military Health Sciences in Hradec Kralove, University of Defence in Brno, and simultaneously she works as a researcher at the Biomedical Research Center and as academic employee at Department of Toxicology and Military Pharmacy, Faculty of Military Health Sciences, University of Defence in Brno.

 

Education

Ph.D. (2014–2021)

University of Defence in Brno, Faculty of Military Health Sciences, study program Toxicology Dissertation title: The development of metod for drugs effecting the central nervous system

Mgr. (2014)

Charles University in Prague, Faculty of Pharmacy, study program Medical bioanalytics Diploma Thesis title: Development of method for in vitro testing of potential drugs Alzheimer’s disease

Bc. (2010)

Charles University in Prague, Faculty of Pharmacy, study program Medical bioanalytics Bachelor Thesis title: In Vitro Inhibitory effect of selected cholinesterase modulators

 

Professional Training 

2018–today

Academic employee, Department of Toxicology and Military Pharmacy, Faculty of Military Health Sciences, University of Defence in Brno

2012–today

Researcher, Biomedical Research Center, University Hospital Hradec Kralove

1996–2018

Technician, Department of Toxicology and Military Pharmacy, Faculty of Military Health Sciences, University of Defence in Brno 

1992–1995

Technician in  EKOS  Hradec Kralove

1991–1992

Technician in Bioanalytika   Hradec Kralove

1987–1990

Technician in Agrochemical laboratory in Hradec Kralove

 

Publication activity

Author or co-author 72 scientific publications with IF

Citation: 660 (excluding self-citations)

H-index: 17

 

Selected publications

2019

Svobodova B, Mezeiova E, Hepnarova V, Hrabinova M, Muckova L, Kobrlova T, Jun D, Soukup O, Jimeno ML, Marco-Contelles J, Korabecny J. Exploring Structure-Activity Relationship in Tacrine-Squaramide Derivatives as Potent Cholinesterase Inhibitors. Biomolecules. 2019 Aug 19;9(8). pii: E379. doi: 10.3390/biom9080379.

Kohelová E, Peřinová R, Maafi N, Korábečný J, Hulcová D, Maříková J, Kučera T, Martínez González L, Hrabinova M, Vorčáková K, Nováková L, De Simone A, Havelek R, Cahlíková L. Derivatives of the β-Crinane Amaryllidaceae Alkaloid Haemanthamine as Multi-Target Directed Ligands for Alzheimer's Disease. Molecules. 2019 Apr 3;24(7). pii: E1307. doi: 10.3390/molecules24071307.

Hepnarova V, Muckova L, Ring A, Pejchal J, Herman D, Misik J, Hrabinova M, Jun D, Soukup O. Pharmacological and toxicological in vitro and in vivo effect of higher doses of oxime reactivators. Toxicol Appl Pharmacol. 2019 Nov 15;383:114776. doi: 10.1016/j.taap.2019.114776.

2018

Kuca K, Jun D, Junova L, Musilek K, Hrabinova M, da Silva JAV, Ramalho TC, Valko M, Wu Q, Nepovimova E, França TCC. Synthesis, Biological Evaluation, and Docking Studies of Novel Bisquaternary Aldoxime Reactivators on Acetylcholinesterase and Butyrylcholinesterase Inhibited by Paraoxon. Molecules.  2018 May 7;23(5). pii: E1103. doi: 10.3390/molecules23051103.

Kuca K, Musilek K, Jun D, Zdarova-Karasova J, Nepovimova E, Soukup O, Hrabinova M, Mikler J, Franca TCC, Da Cunha EFF, De Castro AA, Valis M, Ramalho TC. A newly developed oxime K203 is the most effective reactivator of tabun-inhibited acetylcholinesterase. BMC Pharmacol Toxicol. 2018 Feb 21;19(1):8. doi: 10.1186/s40360-018-0196-3.

Šafratová M, Hošťálková A, Hulcová D, Breiterová K, Hrabcová V, Machado M, Fontinha D, Prudêncio M, Kuneš J, Chlebek J, Jun D, Hrabinová M, Nováková L, Havelek R, Seifrtová M, Opletal L, Cahlíková L. Alkaloids from Narcissus poeticus cv. Pink Parasol of various structural types and their biological activity. Arch Pharm Res. 2018 Feb;41(2):208-218. doi: 10.1007/s12272-017-1000-4. 

2017

Mezeiova E, Korabecny J, Sepsova V, Hrabinova M, Jost P, Muckova L, Kucera T, Dolezal R, Misik J, Spilovska K, Pham NL, Pokrievkova L, Roh J, Jun D, Soukup O, Kaping D, Kuca K. Development of 2-Methoxyhuprine as Novel Lead for Alzheimer's Disease Therapy. Molecules. 2017 Jul 28;22(8). pii: E1265. doi: 10.3390/molecules22081265. 

Jeřábek J, Uliassi E, Guidotti L, Korábečný J, Soukup O, Sepsova V, Hrabinova M, Kuča K, Bartolini M, Peña-Altamira LE, Petralla S, Monti B, Roberti M, Bolognesi ML. Tacrine-resveratrol fused hybrids as multi-target-directed ligands  against Alzheimer's disease. Eur J Med Chem. 2017 Feb 15;127:250-262. Doi 10.1016/j.ejmech.2016.12.048.

2016

Hamulakova S, Poprac P, Jomova K, Brezova V, Lauro P, Drostinova L, Jun D, Sepsova V, Hrabinova M, Soukup O, Kristian P, Gazova Z, Bednarikova Z, Kuca K, Valko M. Targeting copper(II)-induced oxidative stress and the acetylcholinesterase system in Alzheimer's disease using multifunctional tacrine-coumarin hybrid molecules. J Inorg Biochem. 2016 Aug;161:52-62. doi:10.1016/j.jinorgbio.2016.05.001.


  • Introduction
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    • Andrš Martin
    • Benek Ondřej
    • Benková Markéta
    • Doležal Rafael
    • Fabrik Ivo
    • Fabriková Daniela
    • Finger Vladimír
    • Górecki Lukáš
    • Hatlapatková Jana
    • Hrabinová Martina
    • Hympánová Michaela
    • Janoušek Jiří
    • Kobrlová Tereza
    • Konečný Jan
    • Korábečný Jan
    • Kuča Kamil
    • Kupčík Rudolf
    • Lenčo Juraj
    • Maliňák Dávid
    • Marek Jan
    • Marková Aneta
    • Mezeiová Eva
    • Múčková Ľubica
    • Musílek Kamil
    • Novák Martin
    • Prchal Lukáš
    • Psotka Miroslav
    • Pulkrábková Lenka
    • Schmidt Monika
    • Soukup Ondřej
    • Svobodová Barbora
    • Tichý Aleš
    • Vajrychová Marie
    • Vaňousová Andrea
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